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PEN (human)

CAS No. 597578-70-6

PEN (human)( —— )

Catalog No. M30581 CAS No. 597578-70-6

Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    PEN (human)
  • Note
    Research use only, not for human use.
  • Brief Description
    Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
  • Description
    Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
  • In Vitro
    Mouse PEN (mPEN) and rat PEN (rPEN) only differ by one residue at the N-terminal end, whereas human PEN (hPEN) is more divergent and has the sequence PEG instead of PEN.PEN binds and activates a GPCR in the brain.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    GRK (GPCRK)
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    597578-70-6
  • Formula Weight
    2215.49
  • Molecular Formula
    C97H159N27O32
  • Purity
    >98% (HPLC)
  • Solubility
    PBS (pH 7.4):1 mg/mL
  • SMILES
    [H]N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC1=CNC=N1)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)NCC(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)NCC(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C(C)C)C(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Gomes et al (2016) Identification of GPR83 as the receptor for the neuroendocrine peptide PEN. Sci.Signal 9 ra43 PMID:
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